ADCs Cytotoxin with Linkers
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ADCs Cytotoxin with Linkers

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Catalog Product Name CAS Number
BADC-00633 MC-Val-Cit-PAB-duocarmycin 2055896-98-3
MC-Val-Cit-PAB-duocarmycin is a drug-linker conjugate for ADC with potent antitumor activity by using duocarmycin (a DNA minor groove binding alkylating agent), linked via the ADC linker MC-Val-Cit-PAB. Inquiry
BADC-00660 VCP-Eribulin 2130869-17-7
VCP-Eribulin consists the ADCs linker (VCP) and Eribulin. Eribulin is a mechanistically unique microtubule inhibitor for cancer. VCP-Eribulin is an Eribulin-based drug for antibody conjugates. Inquiry
BADC-00666 MAC glucuronide phenol-linked SN-38 2246380-69-6
MAC glucuronide phenol-linked SN-38 is a pH-susceptible lactone MAC glucuronide phenol-linked SN-38 (DNA topoisomerase I inhibitor) drug linker. MAC glucuronide phenol-linked SN-38 is cytotoxic across L540cy cells and Ramos cells with IC50 values of 113 and 67 ng/mL, respectively. Inquiry
BADC-00667 MAC glucuronide α-hydroxy lactone-linked SN-38 2246380-70-9
MAC glucuronide α-hydroxy lactone-linked SN-38 (Topoisomerase I inhibitor) is a stabilized lactone MAC glucuronide α-hydroxy lactone-linked SN-38 drug linker. MAC glucuronide α-hydroxy lactone-linked SN-38 is cytotoxic across L540cy cells and Ramos cells with IC50 values of 99 and 105 ng/mL, respectively. Inquiry
BADC-00668 SC-VC-PAB-DM1 2259318-47-1
SC-VC-PAB-DM1 is a drug-linker conjugate for ADC with with potent antitumor activity by using DM1 (Mertansine, a tubulin inhibitor) , linked via the ADC linker SC-VC-PAB. Inquiry
BADC-00669 Mal-VC-PAB-ABAEP-Azonafide 2259318-48-2
Mal-VC-PAB-ABAEP-Azonafide is a drug-linker conjugate for ADC with with potent antitumor activity by using Azonafide (a cytotoxin), linked via the ADC linker Mal-VC-PAB. Inquiry
BADC-00670 Mal-PEG4-VA-PBD 2259318-50-6
Mal-PEG4-VA-PBD is a drug-linker conjugate for ADC by using the antitumor antibiotic, Pyrrolobenzodiazepine (PBD), linked via Mal-PEG4-VA. Inquiry
BADC-00671 Mal-C2-Gly3-EDA-PNU-159682 2259318-53-9
Mal-C2-Gly3-EDA-PNU-159682, a drug-linker conjugate for ADC, consists a cleavable ADC linker Mal-C2-Gly3-EDA and a potent ADC cytotoxin PNU-159682. Inquiry
BADC-00685 MCC-Modified Daunorubicinol 721945-30-8
Daunorubicinol is a drug-linker conjugate for ADC with potent antitumor activity by using Aur0101 (DNA Topoisomerase II inhibitor), linked via the ADC linker. Inquiry
BADC-00694 MMAF-OMe 863971-12-4
MMAF-Ome is a methoxyl analogue of MMAF, used in antibody-drug conjugates (ADCs) as the antimitotic agent part. The methoxyl works as the reaction group. MMAF is a potent auristatin-derived antineoplastic agent, working by inhibition of tubulin polymerization. It exhibited cytotoxicity in Karpas 299, H3396, 786-O and Caki-1 cells with IC50 values of 119nM, 105nM, 257nM and 200nM after 96-hour treatment. Inquiry
BADC-00696 Val-Cit-PAB-MMAF 863971-56-6
Val-Cit-PAB-MMAF is an antibody drug conjugate cytotoxin. Inquiry
BADC-00704 DBA-DM4 905449-84-5
DBA-DM4 is a drug-linker conjugate composed of a potent a tubulin inhibitor DM1 and a linker SPDP to make antibody drug conjugate (ADC). Inquiry
BADC-00725 OSu-Glu-vc-PAB-MMAE
OSu-Glu-vc-PAB-MMAE is a drug-linker conjugate for ADC by using monomethyl auristatin E (MMAE, a tubulin inhibitor), linked via OSu-Glu-vc-PAB. Inquiry
BADC-00726 OSu-PEG4-vc-PAB-DMEA-Duocarmycin SA
OSu-PEG4-vc-PAB-DMEA-Duocarmycin SA is a drug-linker conjugate for ADC by using Duocarmycin SA (a potent antitumor antibiotic), linked via OSu-PEG4-vc-PAB-DMEA. Inquiry
BADC-00727 Mylotarg-linker
Mylotarg-linker is a drug-linker conjugate for ADC by using N-Acetyl-Calicheamicin and Osu-AcBut-acetyl hydrozide derivative. Inquiry
BADC-00728 OSu-Glu-vc-PAB-MMAD
OSu-Glu-vc-PAB-MMAD is a drug-linker conjugate for ADC by using Monomethyl Dolastatin 10 (MMAD, a potent tubulin inhibitor), linked via OSu-Glu-vc-PAB. Inquiry
BADC-00729 OSu-PEG4-vc-PAB-DMEA-Duocarmycin TM
OSu-PEG4-vc-PAB-DMEA-Duocarmycin TM is a drug-linker conjugate for ADC by using Duocarmycin TM (a potent antitumor antibiotic), linked via OSu-PEG4-vc-PAB-DMEA. Inquiry
BADC-00730 OSu-PEG4-vc-PAB-DMEA-Duocarmycin DM
OSu-PEG4-vc-PAB-DMEA-Duocarmycin DM is a drug-linker conjugate for ADC by using Duocarmycin DM (a potent antitumor antibiotic), linked via OSu-PEG4-vc-PAB-DMEA. Inquiry
BADC-00731 MC-MMD-10
MC-MMD-10 is a drug-linker conjugate for ADC by using MMD-10 and the linker MC. Inquiry
BADC-00732 MA-PEG4-vc-PAB-DMEA-duocarmycin SA
MA-PEG4-vc-PAB-DMEA-duocarmycin SA is a drug-linker conjugate for ADC by using Duocarmycin SA (a potent antitumor antibiotic), linked via MA-PEG4-vc-PAB-DMEA. Inquiry
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